Paolo Tarantino: Ten Reasons to Favor the Gedatolisib Doublet Over the Triplet in Breast Cancer

Paolo Tarantino: Ten Reasons to Favor the Gedatolisib Doublet Over the Triplet in Breast Cancer

Paolo Tarantino, Research Fellow Dana-Farber Cancer Institute and Harvard Medical Schoolpost, shared on LinkedIn:

“Ten reasons why I would favor the newly FDA-approved gedatolisib doublet (fulvestrant/gedatolisib) over the triplet with palbociclib:
  1. VIKTORIA-1 was not designed to compare the two geda arms – yet, the PFS improvement over fulvestrant was similar with or without palbo (HR 0.24, HR 0.33, with overlapping 95%CI)
  2. ORR was also similar, 31% vs 28%, consistent with the idea that palbo does not add much activity
  3. there is no OS advantage from adding palbo, and the current favorable OS trend is similar in both geda arms (HR 0.69 and 0.74)
  4. the PIK3CAmut sub-study of VIKTORIA-1 also confirmed this pattern, with no apparent benefit from the addition of palbo to the doublet
  5. using palbo after prior CDK4/6i has failed to improve outcomes in two randomized trials (PACE, PALMIRA)
  6. the triplet clearly adds toxicity. >50% grade 3 neutropenia (0% without palbo) and higher rates of severe stomatitis and nausea
  7. treatment-related deaths only occurred with the triplet, with two grade 5 toxicities (vs none with the doublet)
  8. the triplet adds logistic burden. A nearly weekly IV infusion and a monthly shot are already burdensome. Adding a third anticancer drug with distinct route of administration and frequent requirement for dose holds further adds complexity.
  9. the triplet further adds costs
  10. we treat this disease to achieve disease control with preservation/improvement of QoL. Adding a third drug which adds toxicity and may worsen QoL, without clear long-term benefit, does not sound like a good deal.”

FDA Approves Gedatolisib – Based Therapy for HR+/HER2− Advanced Breast Cancer Without PIK3CA Mutation

Paolo Tarantino: Ten Reasons to Favor the Gedatolisib Doublet Over the Triplet in Breast Cancer