Matthew Kurian: Trastuzumab Rezetecan Raises New Questions in HER2+ Breast Cancer
Matthew Kurian/ youtube.com

Matthew Kurian: Trastuzumab Rezetecan Raises New Questions in HER2+ Breast Cancer

Matthew Kurian, Executive Committee Member at KYSCO, shared on LinkedIn:

“Another potential challenger in 1L HER2+ metastatic breast cancer first reported by my colleague Paolo Tarantino.

Hengrui announced positive Phase III results for trastuzumab rezetecan (SHR-A1811):

  • SHR-A1811 alone
  • SHR-A1811 + pertuzumab
  • Standard THP

Both SHR-A1811 arms significantly improved PFS vs THP.

The inevitable question: how will this compare with T-DXd?

SHR-A1811 is another HER2-directed topo-I ADC, with a somewhat lower DAR (~6). If it can ultimately deliver T-DXd-like efficacy with meaningfully less ILD/pneumonitis, that could be a real differentiator-especially as we move these ADCs earlier and expose patients for longer periods.

And Hengrui is worth knowing. The emerging model in drug development is increasingly:

Discover/develop in China – rapidly generate clinical proof-of-concept – partner globally.

Hengrui has already built major Western partnerships:

  • GSK: up to 12 programs, $500M upfront + ~$12B potential milestones
  • BMS: 13-program strategic collaboration
  • Merck: $200M upfront + up to $1.77B for global rights to its Lp(a) program

So while many U.S. oncologists may not know Hengrui today, we are likely going to hear this name much more.

For SHR-A1811, I want to see the actual PFS magnitude, ILD rates, CNS activity, whether pertuzumab adds anything – and eventually how it stacks up against T-DXd.”

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Enhertu Plus Pertuzumab Approved in the EU for First-Line HER2-Positive Metastatic Breast Cancer: A New Benchmark After More Than a Decade

Matthew Kurian: Trastuzumab Rezetecan Raises New Questions in HER2+ Breast Cancer