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AMG193 shows antitumor activity in MTAP-deleted solid tumors
Oct 26, 2024, 10:49

AMG193 shows antitumor activity in MTAP-deleted solid tumors

Ben Westphalen, Chair of the Translational Research and Precision Medicine Working Group, shared a recent article by J. Rodon, on X:

Open Access in Annals of Oncology– AMG193, a PRMT5i shows antitumor activity in MTAP-deleted solid tumors with a manageable safety. Important to apply fit for purpose molecular diagnosis to identify patients for clinical trials.”

 

AMG193-solid-tumors

Quoting Pashtoon Kasi ‘s post:

“From a testing standpoint, it could have been easily missed – not all testing platforms cover them.

Especially if testing was a few years ago. Worth repeating testing/knowing coverage of your panel.

Recheck the CDKN2 reports since often co-deleted with MTAP.”

AMG193-solid-tumors

Ben Westphalen reshared his views on X:

“Important point made here – in fact in the trial mentioned above – CDKN2 loss was sufficient for enrollment as the co-deletion is so frequent.”

Peter Brown, Oncology Expert, also shared his views on X:

CDKN2 loss is indeed a significant factor.

I’ve seen this play out in trials where co-deletion is a common occurrence – it’s crucial we consider this in our research design.”

First-in-human study of AMG 193, an MTA-cooperative PRMT5 inhibitor, in patients with MTAP-deleted solid tumors: results from phase I dose exploration

Authors: J. Rodon, H. Prenen, A. Sacher, M. Villalona-Calero, N. Penel, A. El Helali, S. Rottey, N. Yamamoto, F. Ghiringhelli, M.E. Goebeler, T. Doi, S. Postel, Vinay, C.-C. Lin, C. Liu, C.-H. Chuang, K. Keyvanjah, T. Eggert and B.H. O’Neil

AMG193-solid-tumors