Mostafa Faisal: Phase 3 TRANSFORM-1 – Improvments of Adding Navitoclax to Ruxolitinib
Mostafa Faisal and Naveen Pemmaraju

Mostafa Faisal: Phase 3 TRANSFORM-1 – Improvments of Adding Navitoclax to Ruxolitinib

Mostafa Faisal, Adjunct Assistant Professor at Alfaisal University, shared Naveen Pemmaraju’s, Professor in the Department of Leukemia at UT MD Anderson Cancer Center, post on X, adding:

“Phase 3 TRANSFORM-1: Adding navitoclax to ruxolitinib improved spleen responses in JAK inhibitor–naïve intermediate-2/high-risk myelofibrosis.

Results: SVR35 at Week 24: 63.2% vs 31.5% (P<0.0001)
Best Response: Best SVR35 anytime: 76.8% vs 44.1%

Molecular Response: ≥20% VAF reduction: 58.5% vs 45.5%, but symptom improvement was similar (TSS: −10.2 vs −11.6).
Safety: Higher grade 3/4 thrombocytopenia (54% vs 19%), neutropenia (40% vs 9%), and diarrhea (42% vs 17%), with cytopenias generally manageable using dose modifications.”

Quoting Naveen Pemmaraju’s post:

“Proud to share our international randomized frontline Myelofibrosis Ph3 TRANSFORM-1 final results | Navitoclax + RUXO | MPNSM just out in Blood Journals Portfolio today!”

Title: TRANSFORM-1 Phase 3 study: Efficacy and safety of navitoclax plus ruxolitinib in patients with untreated myelofibrosis

Authors: Naveen Pemmaraju, Adam J. Mead, Tim C.P. Somervaille, Francesca Palandri, Steffen Koschmieder, Robert Delage, Jean-Jacques Kiladjian, Christopher B Benton, Srinivas K Tantravahi, Noa Lavi, Su-Peng Yeh, Maria Teresa Gomez Casares, Emanuele Ammatuna, Andrew Bruce McDonald, Sung-Soo Yoon, Keita Kirito, Timothy Devos, Andrew C Perkins, Atanas Radinoff, Omur Gokmen Sevindik, Andrija Bogdanovic, Rastislav Moskal, Jason G. Harb, Bryan C Murray, Qi Jiang, Avijeet S. Chopra, Elektra J. Papadopoulos, Jalaja Potluri, Francesco Passamonti

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